Peptide · Research Monograph · Decapeptide KISS1R/GPR54 agonist

Kisspeptin

Reproductive Hormone Studies

Also known as Kisspeptin-10

Kisspeptin-10 is a ten amino acid peptide. It is the active piece of a longer peptide called kisspeptin-54. It binds a receptor named KISS1R. Studies have measured what happens in the hypothalamus after it binds, and how that signal moves down the reproductive hormone axis. Its discovery changed how the field understood where that signal begins.

Formula
C63H83N17O14
Mol. weight
1302.5 Da
Length
10 residues
CAS
374675-21-5

For laboratory research use only - not for human or animal use

Kisspeptin vial from the Eon Peptides research catalog
Kisspeptin · 10mg · catalog photograph

The molecule, in three dimensions

C63H83N17O141302.5
Drag to turn
Residues · hover to locate10 residues
Heavy atoms
94
Bonds
98
Composition
C63 N17 O14
Rings
4
Metal centre
None
Chain length
10 residues

Every heavy atom is placed from the sequence with ideal bond lengths and angles, so the connectivity is exact. The pose is idealised, an extended chain, and is not a measured conformation. Identity for the lot in stock is confirmed by LC-MS on its certificate.

Molecular data

Molecular formulaC63H83N17O14
Molecular weight1302.5 Da
SequenceTyr-Asn-Trp-Asn-Ser-Phe-Gly-Leu-Arg-Phe-NH2
Sequence length10 residues
CAS / identifier374675-21-5
Physical formWhite lyophilized powder
Available sizes10mg

How it works

  1. GPR54 Agonist

    KISS1R / GPR54 Activation

    Kisspeptin-10 is the shortest active fragment of the KISS1 gene product and binds KISS1R (GPR54) on hypothalamic GnRH neurons - the most potent known endogenous trigger of GnRH neuron activity.

  2. GnRH ↑

    GnRH Pulse Generation

    Receptor activation evokes pulsatile GnRH secretion into the hypophyseal portal circulation, with both the frequency and amplitude of GnRH pulses measured rather than output alone.

  3. LH / FSH ↑

    Gonadotropin Release

    Downstream of GnRH, the pituitary releases luteinizing hormone (robust) and follicle-stimulating hormone (more modest), letting researchers probe upstream control of the gonadal axis.

What the research shows

  1. Reproductive Neuroendocrinology

    GnRH Axis Probing

    Used to evoke discrete LH pulses, enabling characterization of GnRH pulsatility and pituitary responsiveness in controlled models.

  2. Fertility Research

    Gonadotropin Response

    Studied as a stimulus of endogenous LH/FSH to distinguish hypothalamic from pituitary components of reproductive dysfunction.

  3. Development

    Pubertal Signaling

    Investigated for the role of KISS1/GPR54 signaling in the onset and timing of puberty.

Specification

Also Known AsKP-10, Metastin 45-54, Kisspeptin-112-121
TypeDecapeptide - KISS1R/GPR54 agonist
CAS Number374675-21-5
Molecular FormulaC63H83N17O14
Molecular Weight1,302.5 g/mol
Amino Acid SequenceTyr-Asn-Trp-Asn-Ser-Phe-Gly-Leu-Arg-Phe-NH2
Physical AppearanceWhite lyophilized powder
Purity≥99% (HPLC)
Content10 mg per vial

How it's tested

Every lot of Kisspeptin released to the catalog carries a third-party certificate of analysis. 3 documented lots are on file for this compound, with reported HPLC purity from 99.08% to 99.75% (mean 99.52%), issued by Accurate Test Labs and Freedom Diagnostics. 2 of 3 certificates record identity as confirmed.

Documented lots
3
Reported purity
99.08% to 99.75%
Mean purity
99.52%
Issuing labs
Accurate Test Labs, Freedom Diagnostics

All certificates in the COA library →

Frequently asked questions

What is Kisspeptin-10?

Kisspeptin-10 (KP-10) is a synthetic decapeptide corresponding to the C-terminal active fragment of the kisspeptin family encoded by the KISS1 gene. It is a high-affinity agonist of the KISS1R (GPR54) receptor.

How does it differ from Kisspeptin-54?

Kisspeptin-54 is the longer parent peptide; Kisspeptin-10 retains the C-terminal decapeptide that carries full receptor activity, with a shorter sequence and faster in-vivo clearance.

What is GPR54 / KISS1R?

It is the G-protein-coupled receptor for kisspeptins, expressed on GnRH neurons; its activation is essential for normal reproductive-axis function.

How is it stored?

Supplied as a lyophilized powder; store at -20°C, protected from light and moisture. Research use only.

For laboratory research use only. Not a drug, supplement, or medical product; not for human or animal use. All findings referenced are from published preclinical/laboratory research.